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Protein A001920
Automated Data
Not Reviewed
Latest from 7 Sep 2010

Protein kinase C beta

Latest potential protein structures retrieved 7 Sep 2010

Database References

No entries found in this category.

 
Top PDB Blast Hits
PDB IDCompound NameSpeciesE-ValueScoreLinks
2I0EChain A, Structure Of Catalytic Domain Of Human Protein Kinase C Beta Ii Complexed With A Bisindolylmaleimide InhibitorHomo sapiens0.00E0727.242636700999PDBsum
3IW4Chain A, Crystal Structure Of Pkc Alpha In Complex With Nvp-Aeb071Homo sapiens0.00E0617.075557988636PDBsum
2JEDChain A, The Crystal Structure Of The Kinase Domain Of The Protein Kinase C Theta In Complex With Nvp-Xaa228 At 2.32a Resolution.Homo sapiens2.11E-105379.407419647629PDBsum
1XJDChain A, Crystal Structure Of Pkc-Theta Complexed With Staurosporine At 2a ResolutionHomo sapiens2.80E-105379.022220071711PDBsum
3A8WChain A, Crystal Structure Of Pkciota Kinase DomainHomo sapiens1.86E-101366.310634066439PDBsum
3A8XChain A, Crystal Structure Of Pkciota Kinase DomainHomo sapiens1.86E-101366.310634066439PDBsum
1ZRZChain A, Crystal Structure Of The Catalytic Domain Of Atypical Protein Kinase C-IotaHomo sapiens1.04E-100363.999436610935PDBsum
1MRVChain A, Crystal Structure Of An Inactive Akt2 Kinase DomainHomo sapiens4.31E-87318.545886652687PDBsum
1MRYChain A, Crystal Structure Of An Inactive Akt2 Kinase DomainHomo sapiens4.31E-87318.545886652687PDBsum
1GZNChain A, Structure Of Pkb Kinase DomainHomo sapiens1.21E-86317.005088349018PDBsum
1O6LChain A, Crystal Structure Of An Activated AktPROTEIN KINASE B (PKB- Pif Chimera) Ternary Complex With Amp-Pnp And Gsk3 PeptideHomo sapiens1.71E-86316.6198887731PDBsum
1GZKChain A, Molecular Mechanism For The Regulation Of Protein Kinase B Akt By Hydrophobic Motif PhosphorylationHomo sapiens2.07E-86316.234689197183PDBsum
1GZOChain A, Structure Of Protein Kinase B UnphosphorylatedHomo sapiens2.07E-86316.234689197183PDBsum
2JDOChain A, Structure Of Pkb-Beta (Akt2) Complexed With Isoquinoline-5- Sulfonic Acid (2-(2-(4-Chlorobenzyloxy) Ethylamino)ethyl) AmideHomo sapiens2.14E-86316.234689197183PDBsum
2JDRChain A, Structure Of Pkb-Beta (Akt2) Complexed With The Inhibitor A- 443654Homo sapiens2.14E-86316.234689197183PDBsum
2UW9Chain A, Structure Of Pkb-Beta (Akt2) Complexed With 4-(4-Chloro- Phenyl)-4-(4-(1h-Pyrazol-4-Yl)-Phenyl)-PiperidineHomo sapiens2.14E-86316.234689197183PDBsum
2X37Chain A, Structure Of 4-(4-Tert-Butylbenzyl)-1-(7h-Pyrrolo(2,3-D) Pyrimidin-4-Yl)piperidin-4-Amine Bound To PkbHomo sapiens2.14E-86316.234689197183PDBsum
2X39Chain A, Structure Of 4-Amino-N-(4-Chlorobenzyl)-1-(7h-Pyrrolo(2,3-D) Pyrimidin-4-Yl)piperidine-4-Carboxamide Bound To PkbHomo sapiens2.14E-86316.234689197183PDBsum
2XH5Chain A, Structure Of 4-(4-Tert-Butylbenzyl)-1-(7h-Pyrrolo(2,3-D) Pyrimidin-4-Yl)piperidin-4-Amine Bound To PkbHomo sapiens2.14E-86316.234689197183PDBsum
1O6KChain A, Structure Of Activated Form Of Pkb Kinase Domain S474d With Gsk3 Peptide And Amp-PnpHomo sapiens5.78E-86315.079090469431PDBsum
3D0EChain A, Crystal Structure Of Human Akt2 In Complex With Gsk690693Homo sapiens3.50E-85312.382693438009PDBsum
3E87Chain A, Crystal Structures Of The Kinase Domain Of Akt2 In Complex With Atp-Competitive InhibitorsHomo sapiens3.50E-85312.382693438009PDBsum
3E88Chain A, Crystal Structures Of The Kinase Domain Of Akt2 In Complex With Atp-Competitive InhibitorsHomo sapiens3.50E-85312.382693438009PDBsum
3E8DChain A, Crystal Structures Of The Kinase Domain Of Akt2 In Complex With Atp-Competitive InhibitorsHomo sapiens3.50E-85312.382693438009PDBsum
3CQUChain A, Crystal Structure Of Akt-1 Complexed With Substrate Peptide And InhibitorHomo sapiens2.29E-84309.686296406588PDBsum
3CQWChain A, Crystal Structure Of Akt-1 Complexed With Substrate Peptide And InhibitorHomo sapiens2.29E-84309.686296406588PDBsum
3MV5Chain A, Crystal Structure Of Akt-1-Inhibitor ComplexesHomo sapiens2.29E-84309.686296406588PDBsum
3MVHChain A, Crystal Structure Of Akt-1-Inhibitor ComplexesHomo sapiens2.29E-84309.686296406588PDBsum
2R5TChain A, Crystal Structure Of Inactive Serum And Glucocorticoid- Regulated Kinase 1 In Complex With Amp-PnpHomo sapiens2.39E-78289.655918458885PDBsum
3HDMChain A, Crystal Structure Of Serum And Glucocorticoid-Regulated Kinase 1 In Complex With Compound 1Homo sapiens2.39E-78289.655918458885PDBsum
3HDNChain A, Crystal Structure Of Serum And Glucocorticoid-Regulated Kinase 1 In Complex With Compound 2Homo sapiens2.39E-78289.655918458885PDBsum
1A25Chain A, C2 Domain From Protein Kinase C (Beta)Rattus norvegicus3.88E-75278.8703303332PDBsum
3G51Chain A, Structural Diversity Of The Active Conformation Of The N- Terminal Kinase Domain Of P90 Ribosomal S6 Kinase 2Mus musculus1.20E-69260.765950265084PDBsum
3A60Chain A, Crystal Structure Of Unphosphorylated P70s6k1 (Form I)Homo sapiens2.05E-69259.995551113249PDBsum
3A61Chain A, Crystal Structure Of Unphosphorylated P70s6k1 (Form Ii)Homo sapiens2.05E-69259.995551113249PDBsum
3A62Chain A, Crystal Structure Of Phosphorylated P70s6k1Homo sapiens9.03E-69257.684353657745PDBsum
2Z7QChain A, Crystal Structure Of The N-Terminal Kinase Domain Of Human Rsk-1 Bound To Amp-PcpHomo sapiens9.82E-69257.684353657745PDBsum
2Z7RChain A, Crystal Structure Of The N-Terminal Kinase Domain Of Human Rsk1 Bound To StaurosporineHomo sapiens9.82E-69257.684353657745PDBsum
2Z7SChain A, Crystal Structure Of The N-Terminal Kinase Domain Of Human Rsk1 Bound To Purvalnol AHomo sapiens9.82E-69257.684353657745PDBsum
1VZOChain A, The Structure Of The N-Terminal Kinase Domain Of Msk1 Reveals A Novel Autoinhibitory Conformation For A Dual Kinase ProteinHomo sapiens7.10E-64241.505971469216PDBsum
1FOTChain A, Structure Of The Unliganded Camp-Dependent Protein Kinase Catalytic Subunit From Saccharomyces CerevisiaeSaccharomyces cerevisiae1.01E-62237.653975710043PDBsum
1ATPChain E, 2.2 Angstrom Refined Crystal Structure Of The Catalytic Subunit Of Camp-Dependent Protein Kinase Complexed With Mnatp And A Peptide InhibitorMus musculus3.38E-62236.113177406373PDBsum
2QURChain A, Crystal Structure Of F327aK285P MUTANT OF CAMP-Dependent Protein KinaseMus musculus4.24E-62235.727977830456PDBsum
1CDKChain A, Camp-Dependent Protein Kinase Catalytic Subunit (E.C.2.7.1.37) (Protein Kinase A) Complexed With Protein Kinase Inhibitor Peptide Fragment 5-24 (Pki(5-24) Isoelectric Variant Ca) And Mn2+ Adenylyl Imidodiphosphate (Mnamp-Pnp) At Ph 5.6 And 7c And 4cSus scrofa7.99E-62234.572379102704PDBsum
1JBPChain E, Crystal Structure Of The Catalytic Subunit Of Camp- Dependent Protein Kinase Complexed With A Substrate Peptide, Adp And DetergentMus musculus9.92E-62234.572379102704PDBsum
1CTPChain E, Structure Of The Mammalian Catalytic Subunit Of Camp- Dependent Protein Kinase And An Inhibitor Peptide Displays An Open ConformationSus scrofa1.16E-61234.187179526787PDBsum
2ERZChain E, Crystal Structure Of C-Amp Dependent Kinase (Pka) Bound To HydroxyfasudilMus musculus1.28E-61234.187179526787PDBsum
2VO0Chain A, Structure Of Pka-Pkb Chimera Complexed With C-(4-(4- Chlorophenyl)-1-(7h-Pyrrolo(2,3-D)pyrimidin-4-Yl)piperidin- 4-Yl)methylamineBos taurus1.34E-61233.801979950869PDBsum
2JDTChain A, Structure Of Pka-Pkb Chimera Complexed With Isoquinoline-5- Sulfonic Acid (2-(2-(4-Chlorobenzyloxy) Ethylamino)ethyl) AmideBos taurus1.36E-61233.801979950869PDBsum
2JDVChain A, Structure Of Pka-Pkb Chimera Complexed With A-443654Bos taurus1.36E-61233.801979950869PDBsum
2UVXChain A, Structure Of Pka-Pkb Chimera Complexed With 7-AzaindoleBos taurus1.36E-61233.801979950869PDBsum
2UW4Chain A, Structure Of Pka-Pkb Chimera Complexed With 2-(4-(5-Methyl- 1h-Pyrazol-4-Yl)-Phenyl)-EthylamineBos taurus1.36E-61233.801979950869PDBsum
2UW7Chain A, Structure Of Pka-Pkb Chimera Complexed With 4-(4-Chloro- Phenyl)-4-(4-(1h-Pyrazol-4-Yl)-Phenyl)-PiperidineBos taurus1.36E-61233.801979950869PDBsum
1FMOChain E, Crystal Structure Of A Polyhistidine-Tagged Recombinant Catalytic Subunit Of Camp-Dependent Protein Kinase Complexed With The Peptide Inhibitor Pki(5-24) And AdenosineMus musculus1.43E-61233.801979950869PDBsum
1JLUChain E, Crystal Structure Of The Catalytic Subunit Of Camp- Dependent Protein Kinase Complexed With A Phosphorylated Substrate Peptide And DetergentMus musculus1.43E-61233.801979950869PDBsum
1RE8Chain A, Crystal Structure Of Camp-Dependent Protein Kinase Complexed With Balanol Analog 2Mus musculus1.43E-61233.801979950869PDBsum
1REJChain A, Crystal Structure Of Camp-Dependent Protein Kinase Complexed With Balanol Analog 1Mus musculus1.43E-61233.801979950869PDBsum
1REKChain A, Crystal Structure Of Camp-Dependent Protein Kinase Complexed With Balanol Analog 8Mus musculus1.43E-61233.801979950869PDBsum
2QVSChain E, Crystal Structure Of Type Iia Holoenzyme Of Camp-Dependent Protein KinaseMus musculus1.43E-61233.801979950869PDBsum
3FJQChain E, Crystal Structure Of Camp-Dependent Protein Kinase Catalytic Subunit Alpha In Complex With Peptide Inhibitor Pki Alpha (6-25)Mus musculus1.43E-61233.801979950869PDBsum
3IDBChain A, Crystal Structure Of (108-268)riib:c Holoenzyme Of Camp- Dependent Protein KinaseMus musculus1.43E-61233.801979950869PDBsum
3IDCChain A, Crystal Structure Of (102-265)riib:c Holoenzyme Of Camp- Dependent Protein KinaseMus musculus1.43E-61233.801979950869PDBsum
2UVYChain A, Structure Of Pka-Pkb Chimera Complexed With Methyl-(4-(9h- Purin-6-Yl)-Benzyl)-AmineBos taurus1.46E-61233.801979950869PDBsum
2UVZChain A, Structure Of Pka-Pkb Chimera Complexed With C-Phenyl-C-(4-( 9h-Purin-6-Yl)-Phenyl)-MethylamineBos taurus1.46E-61233.801979950869PDBsum
2UW0Chain A, Structure Of Pka-Pkb Chimera Complexed With 6-(4-(4-(4- Chloro-Phenyl)-Piperidin-4-Yl)-Phenyl)-9h-PurineBos taurus1.46E-61233.801979950869PDBsum
2UW3Chain A, Structure Of Pka-Pkb Chimera Complexed With 5-Methyl-4- Phenyl-1h-PyrazoleBos taurus1.46E-61233.801979950869PDBsum
2UW5Chain A, Structure Of Pka-Pkb Chimera Complexed With (R)-2-(4- Chloro-Phenyl)-2-(4-1h-Pyrazol-4-Yl)-Phenyl)-EthylamineBos taurus1.46E-61233.801979950869PDBsum
2UW6Chain A, Structure Of Pka-Pkb Chimera Complexed With (S)-2-(4- Chloro-Phenyl)-2-(4-1h-Pyrazol-4-Yl)-Phenyl)-EthylamineBos taurus1.46E-61233.801979950869PDBsum
2UW8Chain A, Structure Of Pka-Pkb Chimera Complexed With 2-(4-Chloro- Phenyl)-2-Phenyl-EthylamineBos taurus1.46E-61233.801979950869PDBsum
2VNWChain A, Structure Of Pka-Pkb Chimera Complexed With (1-(9h-Purin-6- Yl)piperidin-4-Yl)methanamineBos taurus1.46E-61233.801979950869PDBsum
2VNYChain A, Structure Of Pka-Pkb Chimera Complexed With (1-(9h-Purin-6- Yl)piperidin-4-Yl)amineBos taurus1.46E-61233.801979950869PDBsum
2VO3Chain A, Structure Of Pka-Pkb Chimera Complexed With C-(4-(4- Chlorophenyl)-1-(7h-Pyrrolo(2,3-D)pyrimidin-4-Yl)piperidin- 4-Yl)methylamineBos taurus1.46E-61233.801979950869PDBsum
2VO6Chain A, Structure Of Pka-Pkb Chimera Complexed With 4-(4- Chlorobenzyl)-1-(7h-Pyrrolo(2,3-D)pyrimidin-4-Yl)piperidin- 4-YlamineBos taurus1.46E-61233.801979950869PDBsum
1XH9Chain A, Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And MutantsBos taurus1.52E-61233.801979950869PDBsum
1BKXChain A, A Binary Complex Of The Catalytic Subunit Of Camp-Dependent Protein Kinase And Adenosine Further Defines Conformational FlexibilityMus musculus1.60E-61233.801979950869PDBsum
1BX6Chain A, Crystal Structure Of The Potent Natural Product Inhibitor Balanol In Complex With The Catalytic Subunit Of Camp- Dependent Protein KinaseMus musculus1.60E-61233.801979950869PDBsum
2GNFChain A, Protein Kinase A Fivefold Mutant Model Of Rho-Kinase With Y- 27632Bos taurus1.68E-61233.801979950869PDBsum
2GNGChain A, Protein Kinase A Fivefold Mutant Model Of Rho-KinaseBos taurus1.72E-61233.416780374952PDBsum
2GNHChain A, Pka Five Fold Mutant Model Of Rho-Kinase With H1152pBos taurus1.72E-61233.416780374952PDBsum
2GNIChain A, Pka Fivefold Mutant Model Of Rho-Kinase With Inhibitor Fasudil (Ha1077)Bos taurus1.72E-61233.416780374952PDBsum
2CPKChain E, Crystal Structure Of The Catalytic Subunit Of Cyclic Adenosine Monophosphate-Dependent Protein KinaseMus musculus1.75E-61233.416780374952PDBsum
2QCSChain A, A Complex Structure Between The Catalytic And Regulatory Subunit Of Protein Kinase A That Represents The Inhibited StateMus musculus1.75E-61233.416780374952PDBsum
1APMChain E, 2.0 Angstrom Refined Crystal Structure Of The Catalytic Subunit Of Camp-Dependent Protein Kinase Complexed With A Peptide Inhibitor And DetergentMus musculus1.89E-61233.416780374952PDBsum
1L3RChain E, Crystal Structure Of A Transition State Mimic Of The Catalytic Subunit Of Camp-Dependent Protein KinaseMus musculus1.93E-61233.416780374952PDBsum
2GNJChain A, Pka Three Fold Mutant Model Of Rho-Kinase With Y-27632Bos taurus2.00E-61233.416780374952PDBsum
2GNLChain A, Pka Threefold Mutant Model Of Rho-Kinase With Inhibitor H- 1152pBos taurus2.00E-61233.416780374952PDBsum
2GU8Chain A, Discovery Of 2-Pyrimidyl-5-Amidothiophenes As Novel And Potent Inhibitors For Akt: Synthesis And Sar StudiesHomo sapiens2.10E-61233.416780374952PDBsum
2UZTChain A, Pka Structures Of Akt, Indazole-Pyridine InhibitorsBos taurus2.29E-61233.031580799035PDBsum
2UZUChain E, Pka Structures Of Indazole-Pyridine Series Of Akt InhibitorsBos taurus2.29E-61233.031580799035PDBsum
2UZVChain A, Pka Structures Of Indazole-Pyridine Series Of Akt InhibitorsBos taurus2.29E-61233.031580799035PDBsum
2UZWChain E, Pka Structures Of Indazole-Pyridine Series Of Akt InhibitorsBos taurus2.29E-61233.031580799035PDBsum
2F7EChain E, Pka Complexed With (S)-2-(1h-Indol-3-Yl)-1-(5-Isoquinolin-6- Yl-Pyridin-3-Yloxymethyl-EtylamineBos taurus2.48E-61233.031580799035PDBsum
2F7XChain E, Protein Kinase A Bound To (S)-2-(1h-Indol-3-Yl)-1-[5-((E)-2- Pyridin-4-Yl-Vinyl)-Pyridin-3-Yloxymethyl]-EthylamineBos taurus2.48E-61233.031580799035PDBsum
2F7ZChain E, Protein Kinase A Bound To (R)-1-(1h-Indol-3-Ylmethyl)-2-(2- Pyridin-4-Yl-[1,7]naphtyridin-5-Yloxy)-EhylamineBos taurus2.48E-61233.031580799035PDBsum
2OH0Chain E, Crystal Structure Of Protein Kinase A In Complex With Pyridine-Pyrazolopyridine Based InhibitorsBos taurus2.48E-61233.031580799035PDBsum
2OJFChain E, Crystal Structure Of Protein Kinase A In Complex With Pyridine-Pyrazolopyridine Based InhibitorsBos taurus2.48E-61233.031580799035PDBsum
1CMKChain E, Crystal Structures Of The Myristylated Catalytic Subunit Of Camp-Dependent Protein Kinase Reveal Open And Closed ConformationsSus scrofa2.61E-61233.031580799035PDBsum
1SYKChain A, Crystal Structure Of E230q Mutant Of Camp-Dependent Protein Kinase Reveals Unexpected Apoenzyme ConformationMus musculus2.98E-61232.646381223117PDBsum
3MVJChain A, Human Cyclic Amp-Dependent Protein Kinase Pka Inhibitor CompHomo sapiens3.06E-61232.646381223117PDBsum
1YDRChain E, Structure Of Camp-Dependent Protein Kinase, Alpha-Catalytic Subunit In Complex With H7 Protein Kinase Inhibitor 1-(5- Isoquinolinesulfonyl)-2-MethylpiperazineBos taurus3.65E-61232.646381223117PDBsum
1YDSChain E, Structure Of Camp-Dependent Protein Kinase, Alpha-Catalytic Subunit In Complex With H8 Protein Kinase Inhibitor [n-(2- Methylamino)ethyl]-5-IsoquinolinesulfonamideBos taurus3.65E-61232.646381223117PDBsum
1YDTChain E, Structure Of Camp-Dependent Protein Kinase, Alpha-Catalytic Subunit In Complex With H89 Protein Kinase Inhibitor N-[2- (4-Bromocinnamylamino)ethyl]-5-IsoquinolineBos taurus3.65E-61232.646381223117PDBsum
1SMHChain A, Protein Kinase A Variant Complex With Completely Ordered N- Terminal HelixBos taurus3.74E-61232.646381223117PDBsum
1XHAChain A, Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And MutantsBos taurus3.74E-61232.646381223117PDBsum
1Q61Chain A, Pka Triple Mutant Model Of PkbBos taurus4.76E-61232.2611816472PDBsum
1SZMChain A, Dual Binding Mode Of Bisindolylmaleimide 2 To Protein Kinase A (Pka)Bos taurus5.44E-61231.875982071282PDBsum
3DNDChain A, Camp-Dependent Protein Kinase Pka Catalytic Subunit With Pki-5-24Bos taurus5.63E-61231.875982071282PDBsum
3DNEChain A, Camp-Dependent Protein Kinase Pka Catalytic Subunit With Pki-5-24Bos taurus5.63E-61231.875982071282PDBsum
1DSYChain A, C2 Domain From Protein Kinase C (Alpha) Complexed With Ca2+ And PhosphatidylserineRattus norvegicus6.17E-61231.875982071282PDBsum
1SVHChain A, Crystal Structure Of Protein Kinase A In Complex With Azepane Derivative 8Bos taurus7.73E-61231.490782495365PDBsum
1XH5Chain A, Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And MutantsBos taurus7.73E-61231.490782495365PDBsum
1XH6Chain A, Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And MutantsBos taurus7.73E-61231.490782495365PDBsum
1XH8Chain A, Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And MutantsBos taurus7.73E-61231.490782495365PDBsum
2GFCChain A, Camp-Dependent Protein Kinase Pka Catalytic Subunit With Pki-5-24Bos taurus7.73E-61231.490782495365PDBsum
1U7EChain A, The Crystal Structure Of A Protein Kinase A ComplexMus musculus9.68E-61231.105582919448PDBsum
3FHIChain A, Crystal Structure Of A Complex Between The Catalytic And Regulatory (Ri{alpha}) Subunits Of PkaMus musculus9.68E-61231.105582919448PDBsum
2C1AChain A, Structure Of Camp-Dependent Protein Kinase Complexed With Isoquinoline-5-Sulfonic Acid (2-(2-(4-Chlorobenzyloxy) Ethylamino)ethyl)amideBos taurus1.01E-60231.105582919448PDBsum
2C1BChain A, Structure Of Camp-Dependent Protein Kinase Complexed With (4r,2s)-5'-(4-(4-Chlorobenzyloxy)pyrrolidin-2- Ylmethanesulfonyl)isoquinolineBos taurus1.01E-60231.105582919448PDBsum
2VO7Chain A, Structure Of Pka Complexed With 4-(4-Chlorobenzyl)-1-(7h- Pyrrolo(2,3-D)pyrimidin-4-Yl)piperidin-4-YlamineBos taurus1.01E-60231.105582919448PDBsum
1Q8TChain A, The Catalytic Subunit Of Camp-Dependent Protein Kinase (Pka) In Complex With Rho-Kinase Inhibitor Y-27632Bos taurus1.04E-60231.105582919448PDBsum
1Q8UChain A, The Catalytic Subunit Of Camp-Dependent Protein Kinase In Complex With Rho-Kinase Inhibitor H-1152pBos taurus1.04E-60231.105582919448PDBsum
1STCChain E, Camp-Dependent Protein Kinase, Alpha-Catalytic Subunit In Complex With StaurosporineBos taurus1.04E-60231.105582919448PDBsum
1SVEChain A, Crystal Structure Of Protein Kinase A In Complex With Azepane Derivative 1Bos taurus1.04E-60231.105582919448PDBsum
1SVGChain A, Crystal Structure Of Protein Kinase A In Complex With Azepane Derivative 4Bos taurus1.04E-60231.105582919448PDBsum
1VEBChain A, Crystal Structure Of Protein Kinase A In Complex With Azepane Derivative 5Bos taurus1.04E-60231.105582919448PDBsum
3E8CChain A, Crystal Structures Of The Kinase Domain Of Pka In Complex With Atp-Competitive InhibitorsBos taurus1.04E-60231.105582919448PDBsum
3E8EChain A, Crystal Structures Of The Kinase Domain Of Pka In Complex With Atp-Competitive InhibitorsBos taurus1.04E-60231.105582919448PDBsum
1Q24Chain A, Pka Double Mutant Model Of Pkb In Complex With MgatpBos taurus1.12E-60230.72038334353PDBsum
1Q62Chain A, Pka Double Mutant Model Of PkbBos taurus1.12E-60230.72038334353PDBsum
1Q8WChain A, The Catalytic Subunit Of Camp-Dependent Protein Kinase In Complex With Rho-Kinase Inhibitor Fasudil (Ha-1077)Bos taurus1.14E-60230.72038334353PDBsum
1XH4Chain A, Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And MutantsBos taurus1.14E-60230.72038334353PDBsum
3BWJChain A, Complex Of Pka With The Bisubstrate Protein Kinase Inhibitor Lead Compound Arc-1034Bos taurus1.14E-60230.72038334353PDBsum
2JDSChain A, Structure Of Camp-Dependent Protein Kinase Complexed With A- 443654Bos taurus1.18E-60230.72038334353PDBsum
1XH7Chain A, Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And MutantsBos taurus1.26E-60230.72038334353PDBsum
1RDQChain E, Hydrolysis Of Atp In The Crystal Of Y204a Mutant Of Camp- Dependent Protein KinaseMus musculus1.34E-60230.72038334353PDBsum
1J3HChain A, Crystal Structure Of Apoenzyme Camp-Dependent Protein Kinase Catalytic SubunitMus musculus1.84E-60230.335183767613PDBsum
3GPEChain A, Crystal Structure Analysis Of Pkc (Alpha)-C2 Domain Complexe Ca2+ And Ptdins(4,5)p2Rattus norvegicus4.46E-60228.794385463944PDBsum
2UZPChain A, Crystal Structure Of The C2 Domain Of Human Protein Kinase C Gamma.Homo sapiens2.87E-53206.452810060737PDBsum
3C4XChain A, Crystal Structure Of G Protein Coupled Receptor Kinase 1 Bound To Atp And Magnesium Chloride At 2.9aBos taurus2.58E-50196.437621086886PDBsum
3C4YChain A, Crystal Structure Of Apo Form Of G Protein Coupled Receptor Kinase 1 At 7.51aBos taurus2.58E-50196.437621086886PDBsum
3C4ZChain A, Crystal Structure Of G Protein Coupled Receptor Kinase 1 Bound To Adp And Magnesium Chloride At 1.84aBos taurus2.58E-50196.437621086886PDBsum
3C50Chain A, Crystal Structure Of G Protein Coupled Receptor Kinase 1 Bound To Adp And Magnesium Chloride At 2.6aBos taurus2.58E-50196.437621086886PDBsum
3C51Chain A, Crystal Structure Of G Protein Coupled Receptor Kinase 1 Bound To Adp And Magnesium Chloride At 3.55aBos taurus2.58E-50196.437621086886PDBsum
3C4WChain A, Crystal Structure Of G Protein Coupled Receptor Kinase 1 Bound To Atp And Magnesium Chloride At 2.7aBos taurus2.71E-50196.437621086886PDBsum
2ACXChain A, Crystal Structure Of G Protein Coupled Receptor Kinase 6 Bound To AmppnpHomo sapiens1.03E-49194.511623207299PDBsum
3CIKChain A, Human Grk2 In Complex With Gbetagamma SubunitsHomo sapiens2.92E-47186.422432113035PDBsum
3KRWChain A, Human Grk2 In Complex With Gbetgamma Subunits And Balanol (Soak)Homo sapiens3.18E-47186.037232537117PDBsum
3KRXChain A, Human Grk2 In Complex With Gbetgamma Subunits And Balanol (Co-Crystal)Homo sapiens3.18E-47186.037232537117PDBsum
1OMWChain A, Crystal Structure Of The Complex Between G Protein-Coupled Receptor Kinase 2 And Heterotrimeric G Protein Beta 1 And Gamma 2 SubunitsBos taurus4.44E-47185.6520329612PDBsum
1YM7Chain A, G Protein-Coupled Receptor Kinase 2 (Grk2)Bos taurus4.44E-47185.6520329612PDBsum
2BCJChain A, Crystal Structure Of G Protein-Coupled Receptor Kinase 2 In Complex With Galpha-Q And Gbetagamma SubunitsBos taurus4.44E-47185.6520329612PDBsum
2ESMChain A, Crystal Structure Of Rock 1 Bound To FasudilHomo sapiens1.09E-46184.496434233448PDBsum
2ETKChain A, Crystal Structure Of Rock 1 Bound To HydroxyfasudilHomo sapiens1.09E-46184.496434233448PDBsum
2ETRChain A, Crystal Structure Of Rock I Bound To Y-27632Homo sapiens1.09E-46184.496434233448PDBsum
3D9VChain A, Crystal Structure Of Rock I Bound To H-1152p A Di- Methylated Variant Of FasudilHomo sapiens1.09E-46184.496434233448PDBsum
2V55Chain A, Mechanism Of Multi-Site Phosphorylation From A Rock-I:rhoe Complex StructureHomo sapiens1.50E-46184.111234657531PDBsum
2R7BChain A, Crystal Structure Of The Phosphoinositide-Dependent Kinase- 1 (Pdk-1)catalytic Domain Bound To A Dibenzonaphthyridine InhibitorHomo sapiens5.03E-46182.185236777944PDBsum
3IONChain A, Pdk1 In Complex With Compound 8hHomo sapiens5.03E-46182.185236777944PDBsum
1H1WChain A, High Resolution Crystal Structure Of The Human Pdk1 Catalytic DomainHomo sapiens5.11E-46182.185236777944PDBsum
1UVRChain A, Structure Of Human Pdk1 Kinase Domain In Complex With Bim-8Homo sapiens5.11E-46182.185236777944PDBsum
1UU9Chain A, Structure Of Human Pdk1 Kinase Domain In Complex With Bim-3Spodoptera frugiperda5.60E-46182.185236777944PDBsum
1Z5MChain A, Crystal Structure Of N1-[3-[[5-Bromo-2-[[3-[(1- Pyrrolidinylcarbonyl)amino]phenyl]amino]-4- Pyrimidinyl]amino]propyl]-2,2-Dimethylpropanediamide Complexed With Human Pdk1Homo sapiens6.09E-46181.800037202027PDBsum
2PE0Chain A, Crystal Structure Of Human Phosphoinositide-Dependent Protein Kinase 1 (Pdk1) 5-Hydroxy-3-[1-(1h-Pyrrol-2-Yl)- Eth-(Z)-Ylidene]-1,3-Dihydro-Indol-2-One ComplexHomo sapiens6.09E-46181.800037202027PDBsum
2PE1Chain A, Crystal Structure Of Human Phosphoinositide-Dependent Protein Kinase 1 (Pdk1) {2-Oxo-3-[1-(1h-Pyrrol-2-Yl)-Eth- (Z)-Ylidene]-2,3-Dihydro-1h-Indol-5-Yl}-Urea {bx-517} ComplexHomo sapiens6.09E-46181.800037202027PDBsum
2PE2Chain A, Crystal Structure Of Human Phosphoinositide-Dependent Protein Kinase 1 (Pdk1) 3-{5-[2-Oxo-5-Ureido-1,2-Dihydro- Indol-(3z)-Ylidenemethyl]-1h-Pyrrol-3-Yl}-N-(2-Piperidin-1- Yl-Ethyl)-Benzamide ComplexHomo sapiens6.09E-46181.800037202027PDBsum
2BIYChain A, Structure Of Pdk1-S241a Mutant Kinase DomainHomo sapiens7.20E-46181.800037202027PDBsum
3IOPChain A, Pdk-1 In Complex With The Inhibitor Compound-8iHomo sapiens7.32E-46181.800037202027PDBsum
3H9OChain A, Phosphoinositide-Dependent Protein Kinase 1 (Pdk-1) In Complex With Compound 9Homo sapiens7.38E-46181.800037202027PDBsum
2XCHChain A, Crystal Structure Of Pdk1 In Complex With A Pyrazoloquinazoline InhibitorHomo sapiens7.50E-46181.800037202027PDBsum
1OKYChain A, Structure Of Human Pdk1 Kinase Domain In Complex With StaurosporineHomo sapiens7.70E-46181.414837626109PDBsum
1OKZChain A, Structure Of Human Pdk1 Kinase Domain In Complex With Ucn-01Homo sapiens7.70E-46181.414837626109PDBsum
1UU3Chain A, Structure Of Human Pdk1 Kinase Domain In Complex With Ly333531Homo sapiens7.70E-46181.414837626109PDBsum
1UU7Chain A, Structure Of Human Pdk1 Kinase Domain In Complex With Bim-2Homo sapiens7.70E-46181.414837626109PDBsum
1UU8Chain A, Structure Of Human Pdk1 Kinase Domain In Complex With Bim-1Homo sapiens7.70E-46181.414837626109PDBsum
2F2UChain A, Crystal Structure Of The Rho-Kinase Kinase DomainBos taurus1.07E-45181.029638050192PDBsum
2H9VChain A, Structural Basis For Induced-Fit Binding Of Rho-Kinase To The Inhibitor Y27632Bos taurus1.07E-45181.029638050192PDBsum
2XCKChain A, Crystal Structure Of Pdk1 In Complex With A Pyrazoloquinazoline InhibitorHomo sapiens2.33E-45179.87403932244PDBsum
3HRCChain A, Crystal Structure Of A Mutant Of Human Pdk1 Kinase Domain In Complex With AtpHomo sapiens2.76E-45179.87403932244PDBsum
3HRFChain A, Crystal Structure Of Human Pdk1 Kinase Domain In Complex With An Allosteric Activator Bound To The Pif-PocketHomo sapiens2.76E-45179.87403932244PDBsum
2VD5Chain A, Structure Of Human Myotonic Dystrophy Protein Kinase In Complex With The Bisindoylmaleide Inhibitor Bim ViiiHomo sapiens4.15E-43172.55524738001PDBsum
2JC6Chain A, Crystal Structure Of Human Calmodulin-Dependent Protein Kinase 1dHomo sapiens3.49E-36149.443272824969PDBsum
2ELIChain A, Solution Structure Of The Second Phorbol EstersDIACYLGLYCEROL BINDING DOMAIN OF HUMAN PROTEIN Kinase C Alpha TypeHomo sapiens4.03E-35145.976476641713PDBsum

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